マイクロウェーブ合成文献リスト

マイクロウェーブ合成文献リスト

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Articles and
Published Work
A Novel Polymer Supported Approach to Nucleoside Modification
Bae, Suyeal; Lakshman, Mahesh K.
JOC Article, December 2007
7745_a_novel_polymer_supported_approach_to_nucleoside_modification.pdf (254.7KB)
Microwave synthesis for Everyone
Chemistry in Britain, June 2003
2156.pdf (736.9KB)
Microwave synthesis a new wave of synthetic chemistry
LabPlus International, April/May 2003
2154.pdf (1.2MB)
Mikrobolgebaseret kemi – nue muligheter for hurtigere syntese
og metodeudvikling

(in Danish) Dansk Kemi, 84, nr. 2, 2003
2157.pdf (2.6MB)
Microwave synthesis and knowledge management: A productivity revolution
Current Drug Discovery, February 2003
2155.pdf (975.1KB)
Literature References Parallel Modification of Tropane Alkaloids
Aberler, N. S.; Ganesan, A.; Lambert, J. N.; Saubern, S.; Smith, R. Tetrahedron Letters, 2001, 42, 1975-1977.
Related products:

  • PS-Triphenylphosphine
A Polymer Bound Iminophosphorane Approach for the Synthesis of Quinazolines
Zhang, W.; Mayer, J.P.; Hall, S. E.; Weigel, J. A. J. Comb. Chem. 2001, 3, 255-256
Related products:

  • PS-Triphenylphosphine
Mitsunobu Reaction Modifications Allowing Product Isolation Without Chromatography: Application to a Small Parallel Library
Pelletier, J.C.; Kincaid, S. Tetrahedron Letters, 2000, 41, 797-800.
Related products:

  • PS-Triphenylphosphine
Michael Reactions in Water Using Amphiphilic Resin-Supported Quaternary Ammonium Hydroxides
Shibatomi, K.; Nakahashi, T.; Uozumi, Y. Synlett, 2000, 11, 1643-1645.
Related products:

  • ArgoGel
Mitsunobu Reaction Modifications allowing Product Isolation Without Chromatography: Application to a Small Parallel Library
Pelletier, J. C.; Kincaid, S.; Tetrahedron Letters, 2000, 41, 797-800.
Related products:

  • PS-Triphenylphosphine
Parallel Solution Phase Synthesis of N-substituted 2-pyrazoline Libraries
Bauer, U.; Egner, B. J.; Nilsson, I.; Berghult, M.; Tetrahedron Letters , 2000, 41, 2713-2717.
Related products:

  • PS-DIEA
Oxazoline Synthesis from Hydroxamides by Resin Capture and Ring-Forming Release
Pirrung, M. C.; Tumey, N. L.; J. Comb. Chem. 2000, 2, 675-680.
Related products:

  • PS-TsCl
Facile Solid-Phase Construction of Indole Derivatives Based on a Traceless, Activating Sulfonyl Linker
Zhang, H. C.; Ye, H.; Moretto, A. F.; Brumfield, K.; Maryanoff, B. E.; Organic Letters, 2000, 2, 89-92.
Related products:

  • PS-TsCl
Multistep Solution Phase Parallel Synthesis of Spiperone Analogues
Hansen, H.C.; Olsson, R.; Croston, G.; Anderson, C. M.; Bioorganic and Medicinal Chemistry Letters, 2000, 10, 2435-2439.
Related products:

  • PS-TsCl
Use of Polymer Supported Thiophenol for the Synthesis and Purification of a Benzimidazol-2-one Library
Ermann, M.;Simkovsky, N.M.; Roberts, S. M.; parry, D. M.; Baxter, A. D.; Montana, J.G. Tetrahedron Letters, 2000, 41, 2483-2485.
Related products:

  • PS-Thiophenol
A Convenient and Scalable Procedure for Removing the Fmoc Group in Solution
Sheppeck, J. E.; Kar, H.; Hong, H. Tetrahedron Letters, 2000, 41, 5329-5333.
Related products:

  • PS-Thiophenol
Use of Polymer Supported Thiophenol for the Synthesis and Purification of a Benzimidazol-2-one Library
Ermann M., Simkovsky N.M., Roberts S.M., Parry D.M., Baxter A.D. and Montana J.G, Tetrahedron Letters 41, 2483–2485
Related products:

  • PS-Thiophenol
Synthesis of Enamides Related to the Salicylate Antitumor Macrolides Using Coper-Mediated Vinylic Substitution
Shen R., Porco J.A., Organic Letters, 2000, 2, 9, 1333-1336.
Related products:

  • Quest 210
Polymer-Supported Silyl Cyanide and Silyl Azide: Useful Reagents for Solid-Phase Applications
Missio A., Marchioro C., Rossi T., Panunzio M., Selva S., Seneci P. (GlaxoWellcome Medicines Research Centre, Verona (Italy)) Biotechnology and Bioengineering, 2000, 71, 1, 38-43.
Related products:

  • PS-DES
Kinetic Comparison of Trifluroroacetic Acid Cleavage Reactions of Resin-Bound Carbamates, Ureas, Secondary Amides, and Sulfonamides from Benzyl-, Benzhydryl- and Indole-Based Linkers
Yan, B; Nguyen, N; Liu, L.; Holland, G. Raju, B. J.Comb. Chem. 2000, 2, 66-74.
Related products:

  • PS-Indole-CHO
  • PS-MB-CHO
Synthesis of Highly Substituted 5-(Trifluoromethyl)ketoimadazoles Using a Mixed-Solid/Solution Phase Motif
Hamper, B.; Jerome, K.D.; Yalamanchili, G.; Walker, D.M.; Chott, R.C. Mischke, D.A. Biotechnology and Bioengineering (Combinatorial Chemistry), 2000, 71, 1, 28-37.
Polymer-Supported Silyl Cyanide and Silyl Azide: Useful Reagents for Solid-Phase Applications
Missio, A.; Marchioro, C.; Rossi, T; Panunzio, M.; Selva, S.; Seneci, P. Biotechnology and Bioengineering (Combinatorial Chemistry), 2000, 71, 1, 38-43.
Related products:

  • PS-DES

マイクロウェーブ合成で樹脂に結合した試薬やスカベンジャーを使用した成功例として、以下のような論文が発表されています。

  • Increasing Rates of Reaction: Microwave assisted Organic Synthesis for Combinatorial Chemistry
    Lew, A; Krutzik, P.O.; Hart, M.E.; Chamberlain, A. R.; J. Combi. Chem. 2002, 4, 95-105.
  • Synthesis of 1,3,4-Oxadiazoles Using Polymer-Supported Reagents
    Brain, C.T.;Synlett 2001, 382-384.
  • An Efficient Combination of Microwave Dielectric Heating and the use of Solid-Supported Triphenylphosphine for Wittig Reactionse
    Westman, J.; Org. Lett. 2001, 3(23), 3745-3747.
  • A Polymer Supported Thionating Reagent
    Ley, S.V.; Leach, A.G.; Storer, R.I.; J. Chem. Soc. Perkin Trans 2001, 4, 358-361.
  • Thermal and Microwave Assisted Hydrogenation of Electron-deficient Alkenes Using a Polymer-Supported Hydrogen Donor
    Desai, B.; Danks, T. N.; Tetrahedron Letters, 2001, 42, 5963-5965.
  • A Polymer-Supported [1,3,2] Oxazaphospholidine for the Conversion of Isothiocyanates to Isocyanides and Their Subsequent Use in an Ugi Reaction
    Ley, S. V.; Taylor, S.J.; Bioorg. Med. Chem. Lett. 2002, 12, 1813-1816.
  • Fast Microwave-assisted Preparation of Aryl and Vinyl Nitriles and the corresponding Tetrazoles from Organo-halides
    Alterman, M.; Hallberg, A.; J. Org. Chem. 2000, 65, 7984-7989.
  • Rapid Parallel Synthesis Utilizing Microwave Irradiation
    8. Glass, B.; Combs, A.P.; In High-Throughput Synthesis. Principles and Practices; Sucholeiki, I., Ed.; Marcel Dekker:New York, 2001, pp 123-128.
  • High-Throughput Synthesis of N3-Acylated Dihydropyrimidines Combining Microwave-Assisted Synthesis and Scavenging Techniques
    Dallinger, D.; Gorobets, N. Y.; Kappe, C. O.; Org. Lett, 2003, 5, 1205-1208.